斉藤 毅 / Saito, Tsuyoshi

国際統合睡眠医科学研究機構 助教 / Assistant Professor, University of Tsukuba

関連記事 / Related Articles in COTRE

自然に近い眠りを誘う新たな不眠症治療薬の可能性 〜睡眠誘発物質アデノシンのシグナル伝達経路への新アプローチ〜
麻薬性鎮痛薬による眠気に対する新しい戦略を提示 ~眠気の治療薬としてのオレキシン受容体作動薬の可能性~
ナルコレプシーの病因治療効果を確認 ~目覚めを制御する低分子医薬の新たな効果~

 

論文 / Publication

  1. Structure-Activity Relationship between Thiol Group-Trapping Ability of Morphinan Compounds with a Michael Acceptor and Anti-Plasmodium falciparum Activities Noriki Kutsumura, Yasuaki Koyama, Tsuyoshi Saitoh, Naoshi Yamamoto, Yasuyuki Nagumo, Yoshiyuki Miyata, Rei Hokari, Aki Ishiyama, Masato Iwatsuki, Kazuhiko Otoguro, Satoshi Ōmura, Hiroshi Nagase (2020)
  2. Essential structure of orexin 1 receptor antagonist YNT-707, part V: Structure-activity relationship study of the substituents on the 17-amino group. Tsuyoshi Saitoh, Kazunori Seki, Ryo Nakajima, Naoshi Yamamoto, Noriki Kutsumura, Yasuyuki Nagumo, Yoko Irukayama-Tomobe, Yasuhiro Ogawa, Yukiko Ishikawa, Masashi Yanagisawa, Hiroshi Nagase 30 (3) 126893 - 126893 (2020)
  3. Essential structure of orexin 1 receptor antagonist YNT-707, Part IV: The role of D-ring in 4,5-epoxymorphinan on the orexin 1 receptor antagonistic activity. Saitoh T, Seki K, Nakajima R, Yamamoto N, Kutsumura N, Nagumo Y, Irukayama-Tomobe Y, Ogawa Y, Ishikawa Y, Tanimura R, Yanagisawa M, Nagase H Bioorganic & medicinal chemistry letters 29 (18) 2655 - 2658 (2019)
  4. Essential structure of orexin 1 receptor antagonist YNT-707, Part IV: The role of D-ring in 4,5-epoxymorphinan on the orexin 1 receptor antagonistic activity Saitoh, Tsuyoshi, Seki, Kazunori, Nakajima, Ryo, Yamamoto, Naoshi, Kutsumura, Noriki, Nagumo, Yasuyuki, Irukayama-Tomobe, Yoko, Ogawa, Yasuhiro, Ishikawa, Yukiko, Tanimura, Ryuji, Yanagisawa, Masashi, Nagase, Hiroshi Bioorganic & medicinal chemistry letters 29 (18) 2655 - 2658 (2019)
  5. Electrochemical Pinacol Coupling of Acetophenone Using Boron-Doped Diamond Electrode Nakahara Kenshin, Naba Keisuke, Saitoh Tsuyoshi, Sugai Tomoya, Obata Rika, Nishiyama Shigeru, Einaga Yasuaki, Yamamoto Takashi CHEMELECTROCHEM 6 (16) 4153 - 4157 (2019)
  6. Oxidative Cleavage of the Acyl-Carbon Bond in Phenylacetone with Electrogenerated Superoxide Anions Zhang Yan, Sugai Tomoya, Yamamoto Takashi, Yamamoto Naoshi, Kutsumura Noriki, Einaga Yasuaki, Nishiyama Shigeru, Saitoh Tsuyoshi, Nagase Hiroshi CHEMELECTROCHEM 6 (16) 4194 - 4198 (2019)
  7. Corrigendum to "Enhancing endogenous adenosine A2A receptor signaling induces slow-wave sleep without affecting body temperature and cardiovascular function" [Neuropharmacology 144 (2019) 122-132]. Mustafa Korkutata, Tsuyoshi Saitoh, Yoan Cherasse, Shuji Ioka, Feng Duo, Rujie Qin, Nobuyuki Murakoshi, Shinya Fujii, Xuzhao Zhou, Fumihiro Sugiyama, Jiang-Fan Chen, Hidetoshi Kumagai, Hiroshi Nagase, Michael Lazarus 153 153 - 153 (2019)
  8. A NOVEL REARRANGEMENT REACTION OF MORPHINAN TO ARYLMORPHAN SKELETONS AND THE PHARMACOLOGIES OF ARYLMORPHAN DERIVATIVES Yata Masahiro, Kutsumura Noriki, Nagumo Yasuyuki, Yamamoto Naoshi, Saitoh Tsuyoshi, Ishikawa Yukiko, Irukayama-Tomobe Yoko, Yanagisawa Masashi, Nagase Hiroshi HETEROCYCLES 99 (1) 134 - 144 (2019)
  9. Essential structure of orexin 1 receptor antagonist YNT-707, part III: Role of the 14-hydroxy and the 3-methoxy groups in antagonistic activity toward the orexin 1 receptor in YNT-707 derivatives lacking the 4,5-epoxy ring. Yamamoto N, Ohrui S, Okada T, Saitoh T, Kutsumura N, Nagumo Y, Irukayama-Tomobe Y, Ogawa Y, Ishikawa Y, Watanabe Y, Hayakawa D, Gouda H, Yanagisawa M, Nagase H Bioorganic & medicinal chemistry 27 (8) 1747 - 1758 (2019)
  10. Essential structure of orexin 1 receptor antagonist YNT-707, part III: Role of the 14-hydroxy and the 3-methoxy groups in antagonistic activity toward the orexin 1 receptor in YNT-707 derivatives lacking the 4,5-epoxy ring Yamamoto, Naoshi, Ohrui, Sayaka, Okada, Takahiro, Saitoh, Tsuyoshi, Kutsumura, Noriki, Nagumo, Yasuyuki, Irukayama-Tomobe, Yoko, Ogawa, Yasuhiro, Ishikawa, Yukiko, Watanabe, Yurie, Hayakawa, Daichi, Gouda, Hiroaki, Yanagisawa, Masashi, Nagase, Hiroshi Bioorganic & medicinal chemistry 27 (8) 1747 - 1758 (2019)

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※上記の論文リストは researchmapから取得した論文リストにDOIリンク等の情報を付加したものです。筑波大学研究者総覧(TRIOS)または researchmapの論文リストが更新されると後日反映されます。

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知財 / Intellectual properties

  1. 特願2017-202225 : 新規徐波睡眠誘導剤 ラザルス ミハエル, 斉藤 毅, 長瀬 博, コルクタタ ムスタファ, 井岡 秀二
  2. JP2017012607 : 骨代謝調節用組成物 禹 済泰, 車 炳允, 岩井 みどり, 米澤 貴之, 鄭 雄一, 西山 繁, 斉藤 毅
  3. JP2016081995 : モルヒナン誘導体及びその医薬用途 長瀬 博, 山本 直司, 入鹿山 容子, 斉藤 毅, 柳沢 正史, 南雲 康行
  4. 特願2012-265382 : 環化化合物の製造方法、及び、環化化合物を含有する溶液の発光方法 斉藤 毅, 西山 繁, 井岡 秀二, 牧 昌次郎, 丹羽 治樹
  5. JP2016067405 : スルホンアミド誘導体またはその薬学的に許容される酸付加塩 長瀬 博, 柳沢 正史, 斉藤 毅, 沓村 憲樹, 入鹿山 容子
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発行:筑波大学 URA研究戦略推進室・研究推進部